SCHEMBL7423501

SCHEMBL7423501

N#Cc1cc(-n2cncn2)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP2A6 P11509 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
FBP1 P09467 1/20 0.35
DPP4 P27487 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP19A1 P11511 6/20 0.34
HTR1A P08908 1/20 0.34
HTR2C P28335 1/20 0.34
CHRNA7 P36544 1/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6592711 0.80 SMN1; SMN2 (0.50) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL2075610 0.78 S1PR3 (0.43) KDM4EALDH1A1SMN1; SMN2CYP2A6
SCHEMBL10676226 0.76 ADORA2A (0.35) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL7473254 0.76 FBP1 (0.46) KDM4EALDH1A1SMN1; SMN2CYP1A2CYP2C9
SCHEMBL1852173 0.76 SMN1; SMN2 (0.46) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL6225101 0.76 KDM4E (0.46) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL356291 0.76 ALDH1A1 (0.46) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL1824296 0.76 KDM4E (0.46) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL2270763 0.73 KDM4E (0.55) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2
SCHEMBL3313764 0.72 KDM4E (0.50) KDM4EALDH1A1SMN1; SMN2CYP2A6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691967-B1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS EISAI CO LTD (JP) 1998-09-02 EP disclosed
US-5707998-A CYCLIC-GMP PHOSPHODIESTERASE INHIBITORS, TREATING CARDIOVASCULAR DISORDERS AND ASTHMA EISAI CO., LTD. (JP) 1998-01-13 US disclosed
WO-1994022855-A1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS EISAI CO., LTD. (JP) 1994-10-13 WO disclosed