SCHEMBL7423540

SCHEMBL7423540

CCCn1c(=O)[nH]c(=S)c2[nH]c(C(C)C)nc21

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423089 0.89 ADORA2A (0.39) ADORA2AADORA2B
SCHEMBL8000439 0.86 ADORA2A (0.41) ADORA2AADORA2B
SCHEMBL5226057 0.86 ADORA2A (0.56) ADORA2AADORA2B
SCHEMBL7274376 0.83 ADORA2A (0.68) ADORA2AADORA2B
SCHEMBL7425894 0.83 ADORA2A (0.53) ADORA2AADORA2B
SCHEMBL9706669 0.81 ADORA2A (0.45) ADORA2AADORA2B
SCHEMBL7673623 0.80 TLR7 (0.41) ADORA2AADORA2B
SCHEMBL7420292 0.80 ADORA1 (0.44) ADORA2AADORA2B
SCHEMBL9788499 0.78 KDM4E (0.33)
SCHEMBL5231243 0.78 PDE2A (0.46) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6268373-B1 ENZYME INHIBITORS EURO-CELTIQUE S.A. (LU) 2001-07-31 US disclosed
US-6025361-A EFFECTIVE PDE IV INHIBITORS, ASTHMA EURO-CELTIQUE, S.A. (LU) 2000-02-15 US disclosed
US-5977119-A Trisubstituted thioxanthines EURO-CELTIQUE, S.A. (LU) 1999-11-02 US disclosed
EP-0799040-A4 TRISUBSTITUTED THIOXANTHINES EURO CELTIQUE SA (LU) 1998-04-01 EP disclosed
EP-0799040-A1 TRISUBSTITUTED THIOXANTHINES Euroceltique S.A. (LU) 1997-10-08 EP disclosed
WO-1996018400-A1 TRISUBSTITUTED THIOXANTHINES EURO-CELTIQUE, S.A. (LU) 1996-06-20 WO disclosed