SCHEMBL9706669

SCHEMBL9706669

CCCn1c(=O)[nH]c(=S)c2[nH]c(C)nc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.45
ADORA2B P29275 4/20 0.45
ADORA1 P30542 2/20 0.45
PDE4A P27815 3/20 0.44
PDE4B Q07343 3/20 0.44
PDE4C Q08493 3/20 0.44
PDE4D Q08499 3/20 0.44
HPGD P15428 2/20 0.44
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
SIRT5 Q9NXA8 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
BLM P54132 1/20 0.44
PDE3A Q14432 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PDE2A O00408 1/20 0.43
PDE1A P54750 1/20 0.43
PDE1B Q01064 1/20 0.43
PDE1C Q14123 1/20 0.43
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419694 0.91 PDE4A (0.47) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9706609 0.88 HPGD (0.49) ADORA2AADORA2BADORA1PDE4APDE4B
SCHEMBL7420292 0.84 ADORA1 (0.44) ADORA2AADORA2BADORA1PDE4APDE4B
SCHEMBL5231243 0.81 PDE2A (0.46) ADORA2AADORA2BADORA1PDE4APDE4B
SCHEMBL7423540 0.81 ADORA2A (0.45) ADORA2AADORA2B
SCHEMBL1460912 0.81 PDE1A (0.58) HPGDSIRT1SIRT3SIRT5BLM
SCHEMBL5233098 0.80 ADORA1 (0.48) ADORA2AADORA2BADORA1
SCHEMBL7425220 0.79 ADORA1 (0.69) ADORA2AADORA2BADORA1ADORA3
SCHEMBL9645587 0.79 ADORA1 (0.50) ADORA2AADORA2BADORA1
SCHEMBL7866628 0.79 ADORA2B (0.61) ADORA2AADORA2BADORA1ADORA3HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4710503-A 6-thioxanthine derivatives EUROCELTIQUE S.A. (LU) 1987-12-01 US claimed
EP-0191313-B1 6-THIOXANTHINE DERIVATIVES Euro-Celtique S.A. (LU) 1992-10-28 EP disclosed
US-4820709-A 6-thioxanthine derivatives EUROCELTIQUE, S.A. (LU) 1989-04-11 US disclosed
US-4710503-A 6-thioxanthine derivatives EUROCELTIQUE S.A. (LU) 1987-12-01 US disclosed
EP-0191313-A1 6-Thioxanthine derivatives Euro-Celtique S.A. (LU) 1986-08-20 EP disclosed