SCHEMBL7424186

SCHEMBL7424186

Cc1cc(CO)c(C(C)C)c(-c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.46
CD274 Q9NZQ7 1/20 0.46
NUDT1 P36639 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
METAP2 P50579 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
PTGS1 P23219 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ESR2 Q92731 1/20 0.36
BACE1 P56817 1/20 0.35
GCGR P47871 1/20 0.35
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24469036 0.80 SHBG (0.33)
SCHEMBL7418616 0.79 BACE1 (0.47) NUDT1PTGDR2METAP2HDAC7ESR2
SCHEMBL10014387 0.77 PDCD1 (0.50) PDCD1CD274PTGDR2METAP2HDAC7
SCHEMBL26651931 0.74 SHBG (0.34)
SCHEMBL9485214 0.73 PDCD1 (0.53) PDCD1CD274PTGDR2HDAC7PTGS1
SCHEMBL14194630 0.73 PDCD1 (0.53) PDCD1CD274PTGDR2HDAC7PTGS1
SCHEMBL22380329 0.73 ALOX15 (0.33)
SCHEMBL30306137 0.71 BACE1 (0.41) PDCD1CD274PTGDR2METAP2HDAC7
SCHEMBL28221505 0.70 PDCD1 (0.46) PDCD1CD274ESR2BACE1
SCHEMBL21670389 0.69 HDAC7 (0.45) NUDT1PTGDR2METAP2HDAC7PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002022584-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-03-21 WO disclosed