SCHEMBL7424336

SCHEMBL7424336

COC(=O)c1ccc(CS(=O)(=O)NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.50
MAPT P10636 2/20 0.50
MEN1 O00255 2/20 0.50
LMNA P02545 2/20 0.50
KMT2A Q03164 2/20 0.50
GAA P10253 1/20 0.50
KDM4E B2RXH2 3/20 0.49
RAB9A P51151 2/20 0.49
TSHR P16473 1/20 0.49
ALDH1A1 P00352 2/20 0.48
HPGD P15428 2/20 0.48
HTT P42858 2/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CRHBP P24387 1/20 0.48
CYP2C19 P33261 1/20 0.48
CRHR2 Q13324 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NOD2 Q9HC29 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3916464 0.82 POLB (0.62) POLBMAPTKDM4ERAB9ATSHR
SCHEMBL18424863 0.80 CA1 (0.60) POLBMAPTMEN1KMT2AKDM4E
SCHEMBL3850206 0.80 POLB (0.72) POLBMAPTLMNATSHRALDH1A1
SCHEMBL24360900 0.80 CA1 (0.57) LMNAKMT2AKDM4EALDH1A1HPGD
SCHEMBL19165774 0.76 HPGD (0.63) POLBMAPTLMNAKMT2ARAB9A
SCHEMBL27556687 0.75 LOXL2 (0.61) MAPTMEN1KMT2AKDM4ETSHR
SCHEMBL21761420 0.75 ALDH1A1 (0.69) POLBMAPTMEN1LMNAKMT2A
SCHEMBL7318888 0.75 FLT1 (0.58) POLBMEN1LMNAKMT2AKDM4E
SCHEMBL119461 0.74 POLB (0.72) POLBMAPTLMNAGAATSHR
SCHEMBL709955 0.74 LOXL2 (0.59) MAPTMEN1KMT2ATSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0960104-A1 N-(AMIDINOPHENYL)-N'-(SUBST.)-3H-2,4-BENZODIAZEPIN-3-ONE DERIVATIVES AS FACTOR XA INHIBITORS Du Pont Pharmaceuticals Company (US) 1999-12-01 EP disclosed
WO-1997038984-A1 N-(AMIDINOPHENYL)-N'-(SUBST.)-3H-2,4-BENZODIAZEPIN-3-ONE DERIVATIVES AS FACTOR XA INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1997-10-23 WO disclosed