SCHEMBL7424618

SCHEMBL7424618

Cc1cc(C(=O)O)cc(-c2cnccc2C(C)C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 2/20 0.53
F2 P00734 1/20 0.49
TPMT P51580 1/20 0.42
HCAR2 Q8TDS4 1/20 0.41
LDHA P00338 1/20 0.40
LDHB P07195 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
KMO O15229 1/20 0.38
HCAR1 Q9BXC0 1/20 0.38
CTRC Q99895 1/20 0.36
CYP11B2 P19099 1/20 0.36
MAPT P10636 1/20 0.36
GSK3B P49841 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
XDH P47989 1/20 0.36
SYK P43405 1/20 0.36
CNR2 P34972 1/20 0.35
DHODH Q02127 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423958 0.86 RPS6KA3 (0.50) RPS6KA3F2CYP11B2MAPTGSK3B
SCHEMBL29236274 0.83 TPMT (0.47) TPMTHCAR2RXRARXRBKMO
SCHEMBL31027177 0.83 TPMT (0.47) TPMTHCAR2RXRARXRBKMO
SCHEMBL7422808 0.80 TPMT (0.47) TPMTLDHALDHBRXRARXRB
SCHEMBL14395132 0.73 KMO (0.67) TPMTHCAR2RXRARXRBKMO
SCHEMBL6910260 0.71 RPS6KA3 (0.57) RPS6KA3GSK3BSLC22A12
SCHEMBL15521802 0.70 TPMT (0.64) TPMTHCAR2RXRARXRBHCAR1
SCHEMBL21105124 0.70 RPS6KA3 (0.60) RPS6KA3MAPTGSK3BSLC22A12
SCHEMBL28270190 0.70 KDM4C (0.49) HCAR2KMOMAPTDHODHSLC22A12
SCHEMBL17231196 0.70 TPMT (0.76) TPMTHCAR2RXRARXRBHCAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002022584-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-03-21 WO disclosed