SCHEMBL7423958

SCHEMBL7423958

COC(=O)c1cc(C)cc(-c2cnccc2C(C)C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 1/20 0.50
F2 P00734 1/20 0.49
ATM Q13315 1/20 0.44
CNR2 P34972 2/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP46A1 Q9Y6A2 1/20 0.41
SLC2A1 P11166 1/20 0.41
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
FGFR1 P11362 1/20 0.38
SRC P12931 1/20 0.38
FGFR2 P21802 1/20 0.38
FGFR4 P22455 1/20 0.38
FGFR3 P22607 1/20 0.38
TGFBR1 P36897 1/20 0.37
NEK1 Q96PY6 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424618 0.86 RPS6KA3 (0.53) RPS6KA3F2CNR2CYP11B2MAPT
SCHEMBL7419776 0.82 CNR2 (0.46) CNR2SLC7A5TDP1
SCHEMBL21711900 0.72 WDR5 (0.47) ATMALDH1A1CYP46A1SLC2A1CYP2A6
SCHEMBL12261518 0.70 KDM4E (0.56) ATMALDH1A1CYP46A1TGFBR1KDM4E
SCHEMBL21712000 0.69 LOXL2 (0.47) SLC2A1CYP2A6
SCHEMBL31027179 0.69 GPBAR1 (0.56) SLC2A1
SCHEMBL29236310 0.69 GPBAR1 (0.56) SLC2A1
SCHEMBL31027177 0.69 TPMT (0.47) CNR2CYP11B1CYP11B2
SCHEMBL30571537 0.69 SLC6A3 (0.56) ATMCNR2ALDH1A1CYP46A1KDM4E
SCHEMBL29236274 0.69 TPMT (0.47) CNR2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002022584-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-03-21 WO disclosed