SCHEMBL7424626

SCHEMBL7424626

COC(=O)[C@H](CC(C)C)NC(=O)c1ccc(OC)c(OC2CCCC2)c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 10/20 0.66
PDE4B Q07343 10/20 0.66
PDE4C Q08493 10/20 0.66
PDE4D Q08499 10/20 0.66
TAS1R3 Q7RTX0 6/20 0.65
TAS1R1 Q7RTX1 6/20 0.65
BCL2L1 Q07817 2/20 0.56
EPHX2 P34913 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323597 1.00 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DTAS1R3
SCHEMBL19083995 0.87 TAS1R3 (0.62) PDE4APDE4BPDE4CPDE4DTAS1R3
SCHEMBL7450501 0.83 PDE4D (0.75) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL202816 0.82 PDE4D (0.74) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL7512973 0.82 PDE4D (0.74) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL7424332 0.81 PDE4D (0.60) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL703468 0.79 TAS1R3 (1.00) TAS1R3TAS1R1BCL2L1
SCHEMBL703467 0.79 TAS1R3 (1.00) TAS1R3TAS1R1BCL2L1
SCHEMBL700708 0.79 TAS1R3 (1.00) TAS1R3TAS1R1BCL2L1
SCHEMBL700709 0.79 TAS1R3 (1.00) TAS1R3TAS1R1BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998056756-A1 CATECHOL AMINO ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CHEIL JEDANG CORPORATION (KR) 1998-12-17 WO claimed
EP-2193808-A1 Synergistic combination Nycomed GmbH (DE) 2010-06-09 EP disclosed
WO-1998056756-A1 CATECHOL AMINO ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CHEIL JEDANG CORPORATION (KR) 1998-12-17 WO disclosed