SCHEMBL7424627

SCHEMBL7424627

CCOC(=O)C1CCN(c2nc(NCc3ccc4c(c3)OOC4)c3cc(N(C)C)ccc3n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4C Q08493 2/20 0.48
PDE4D Q08499 2/20 0.48
PDE2A O00408 1/20 0.47
PDE5A O76074 1/20 0.47
PDE1A P54750 1/20 0.47
PDE1B Q01064 1/20 0.47
PDE1C Q14123 1/20 0.47
KDM4E B2RXH2 1/20 0.42
CTNNB1 P35222 10/20 0.41
TCF7L2 Q9NQB0 10/20 0.41
HRH4 Q9H3N8 3/20 0.41
BRD4 O60885 2/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
SHMT2 P34897 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418631 0.87 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL6031648 0.79 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL9095949 0.79 PDE4A (0.73) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL7471242 0.78 PDE4A (0.77) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL7797879 0.77 SHMT2 (0.46) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL4931286 0.77 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL5598718 0.77 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DPDE2A
Hydrochloric Acid SCHEMBL8610408 0.76 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE2A
Hydrochloric Acid SCHEMBL7503522 0.76 PDE4A (0.79) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL7495905 0.75 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994022855-A1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS EISAI CO., LTD. (JP) 1994-10-13 WO disclosed