SCHEMBL742472

SCHEMBL742472

COc1cccc(CNc2nc(SCc3ccccc3)nc3nc[nH]c23)c1O.Clc1nc(SCc2ccccc2)nc2nc[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
TSHR P16473 2/20 0.48
TP53 P04637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
STAT3 P40763 1/20 0.43
IP6K1 Q92551 1/20 0.42
CXCR2 P25025 1/20 0.41
CDK1 P06493 2/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
TMIGD3 P0DMS9 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
HTT P42858 3/20 0.40
LMNA P02545 3/20 0.40
ALOX15 P16050 1/20 0.40
MAPT P10636 4/20 0.40
ALDH1A1 P00352 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL774658 0.95 SMN1; SMN2 (0.53) SMN1; SMN2TSHRTP53HSD17B10STAT3
SCHEMBL742471 0.78 CCNE1 (0.45) SMN1; SMN2TSHRTP53CDK1HTT
SCHEMBL741057 0.77 PIN1 (0.56) SMN1; SMN2TSHRHSD17B10CXCR2CDK1
SCHEMBL30411673 0.74 SMN1; SMN2 (0.80) SMN1; SMN2TSHRTP53HSD17B10HTT
SCHEMBL4924809 0.74 SMN1; SMN2 (0.80) SMN1; SMN2TSHRTP53HSD17B10HTT
Chloroform SCHEMBL743258 0.74 PIN1 (0.53) SMN1; SMN2TSHRHSD17B10CXCR2CDK1
SCHEMBL30523415 0.72 HSD17B10 (0.69) SMN1; SMN2TSHRTP53HSD17B10STAT3
SCHEMBL16146326 0.72 HSD17B10 (0.69) SMN1; SMN2TSHRTP53HSD17B10STAT3
SCHEMBL3907002 0.70 CDK1 (0.48) TSHRHSD17B10STAT3IP6K1CXCR2
SCHEMBL16146477 0.70 SMN1; SMN2 (0.56) SMN1; SMN2TSHRTP53HSD17B10STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430036-A1 SUBSTITUTED 6-(BENZYLAMINO) PURINE RIBOSIDE DERIVATIVES, USE THEREOF AND COMPOSITIONS CONTAINING THESE DERIVATIVES Univerzita Palackého v Olomouci (CZ) 2012-03-21 EP disclosed
WO-2010130233-A1 SUBSTITUTED 6-(BENZYLAMINO) PURINE RIBOSIDE DERIVATIVES, USE THEREOF AND COMPOSITIONS CONTAINING THESE DERIVATIVES UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2010-11-18 WO disclosed