SCHEMBL7424743

SCHEMBL7424743

COC(=O)[C@H](Cc1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1)NC(=O)[C@H]1CSCN1S(=O)(=O)c1cccc2c(N(C)C)cccc12

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 19/20 0.43
ITGB1 P05556 18/20 0.43
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428679 0.93 ITGA4 (0.51) ITGA4ITGB1
SCHEMBL7429058 0.86 ITGA4 (0.56) ITGA4ITGB1CYP3A4
SCHEMBL7422799 0.85 ITGB1 (0.48) ITGA4ITGB1
SCHEMBL7423777 0.81 ITGB1 (0.51) ITGA4ITGB1
SCHEMBL7426191 0.78 ITGA4 (0.65) ITGA4ITGB1
SCHEMBL6742321 0.78 ITGB1 (0.50) ITGA4ITGB1
SCHEMBL6739377 0.78 ITGB1 (0.50) ITGA4ITGB1
SCHEMBL7428465 0.78 ITGB1 (0.58) ITGA4ITGB1
SCHEMBL6740760 0.78 ITGA4 (0.48) ITGA4ITGB1
SCHEMBL6744310 0.78 ITGA4 (0.48) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089989-A1 INHIBITORS OF ALPHA4BETA1 MEDIATED CELL ADHESION PHARMACIA & UPJOHN COMPANY (US) 2001-04-11 EP disclosed
WO-1999067230-A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION PHARMACIA & UPJOHN COMPANY (US) 1999-12-29 WO disclosed