SCHEMBL7424976

SCHEMBL7424976

COc1cc(CC(=O)Nc2ccc(C(CC(=O)O)NS(=O)(=O)C3=NCN(C)C3)cn2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 15/20 0.55
ITGB1 P05556 14/20 0.55
CHEK1 O14757 1/20 0.38
ITGB3 P05106 3/20 0.38
ITGAV P06756 3/20 0.38
P2RX7 Q99572 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649474 0.89 ITGB1 (0.54) ITGA4ITGB1
SCHEMBL7645880 0.89 ITGA4 (0.49) ITGA4ITGB1ITGB3ITGAV
SCHEMBL7648770 0.88 ITGA4 (0.58) ITGA4ITGB1
SCHEMBL7425612 0.88 ITGA4 (0.53) ITGA4ITGB1CHEK1P2RX7
SCHEMBL7387358 0.88 ITGA4 (0.62) ITGA4ITGB1CHEK1P2RX7
SCHEMBL7391722 0.85 ITGB1 (0.57) ITGA4ITGB1ITGB3ITGAV
SCHEMBL7424964 0.84 ITGA4 (0.55) ITGA4ITGB1CHEK1
SCHEMBL7588934 0.83 ITGA4 (0.60) ITGA4ITGB1CHEK1P2RX7
SCHEMBL7647038 0.83 ITGA4 (0.47) ITGA4ITGB1CHEK1ITGB3ITGAV
SCHEMBL7561313 0.83 ITGB1 (0.63) ITGA4ITGB1CHEK1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479519-B1 INHIBITORS OF CELL ADHESION; TREATMENT OF ASTHMA OR INFLAMMATORY BOWEL DISEASE AVENTIS PHARMA LIMITED (GB) 2002-11-12 US disclosed
EP-1027328-A1 SUBSTITUTED ANILIDES Aventis Pharma Limited (GB) 2000-08-16 EP disclosed
WO-1999023063-A1 SUBSTITUTED ANILIDES AVENTIS PHARMA LIMITED (GB) 1999-05-14 WO disclosed