SCHEMBL7425399

SCHEMBL7425399

COc1cc(C(CC2CCN(C(CC(=O)O)c3ccc(OC)c(OC)c3)CC2)NC(C)=O)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 9/20 0.46
ITGA4 P13612 9/20 0.46
TNF P01375 1/20 0.41
POLB P06746 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424846 0.95 ITGB1 (0.45) ITGB1ITGA4TNFPOLBPDE4A
SCHEMBL7425026 0.95 ITGB1 (0.47) ITGB1ITGA4L3MBTL1ALDH1A1MAPT
SCHEMBL7535883 0.91 ITGA4 (0.46) ITGB1ITGA4L3MBTL1ALDH1A1MAPT
SCHEMBL7428883 0.91 ITGB1 (0.50) ITGB1ITGA4L3MBTL1ALDH1A1MAPT
SCHEMBL7483888 0.88 ITGA4 (0.49) ITGB1ITGA4L3MBTL1ALDH1A1MAPT
SCHEMBL7393051 0.88 ITGB1 (0.47) ITGB1ITGA4TNFPDE4APDE4B
SCHEMBL7431427 0.86 ITGB1 (0.53) ITGB1ITGA4POLBL3MBTL1MAPT
SCHEMBL7430152 0.85 ITGA4 (0.48) ITGB1ITGA4L3MBTL1ALDH1A1MAPT
SCHEMBL7425440 0.84 ITGB1 (0.44) ITGB1ITGA4MEN1KMT2A
SCHEMBL7425213 0.83 ITGB1 (0.49) ITGB1ITGA4TNFPOLBPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed