SCHEMBL7425546

SCHEMBL7425546

COC(=O)CC(NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)C(C)C)C(=O)C=[N+]=[N-]

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.54
REN P00797 7/20 0.48
BACE1 P56817 2/20 0.45
BACE2 Q9Y5Z0 2/20 0.45
OPRD1 P41143 1/20 0.45
CASP3 P42574 2/20 0.41
CASP7 P55210 1/20 0.41
CASP9 P55211 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418200 0.91 CASP1 (0.62) CASP1RENBACE1BACE2OPRD1
SCHEMBL7420728 0.87 CASP1 (0.57) CASP1RENBACE1BACE2OPRD1
SCHEMBL7416737 0.84 CASP1 (0.53) CASP1RENBACE1BACE2OPRD1
SCHEMBL5081623 0.83 CASP1 (0.60) CASP1RENBACE1BACE2OPRD1
SCHEMBL7296792 0.80 CASP1 (0.55) CASP1RENBACE1BACE2OPRD1
SCHEMBL5689768 0.78 CASP1 (0.59) CASP1RENBACE1BACE2OPRD1
SCHEMBL27825824 0.78 CASP1 (0.67) CASP1BACE1BACE2OPRD1CASP3
SCHEMBL9241543 0.78 CASP1 (0.67) CASP1BACE1BACE2OPRD1CASP3
SCHEMBL14370014 0.77 CASP1 (0.60) CASP1RENBACE1BACE2OPRD1
SCHEMBL2314756 0.76 CASP1 (0.61) CASP1BACE1BACE2OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014777-A1 PEPTIDYL DERIVATIVES AS INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME MERCK & CO., INC. (US) 1993-08-05 WO disclosed