SCHEMBL7416737

SCHEMBL7416737

CC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](C)C(=O)NC(CC(=O)O)C(=O)C=[N+]=[N-])C(C)C

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.53
BACE1 P56817 5/20 0.50
BACE2 Q9Y5Z0 2/20 0.50
ACE P12821 1/20 0.47
REN P00797 1/20 0.45
OPRD1 P41143 1/20 0.45
CASP3 P42574 1/20 0.44
CASP7 P55210 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418200 0.93 CASP1 (0.62) CASP1BACE1BACE2RENOPRD1
SCHEMBL7420728 0.88 CASP1 (0.57) CASP1BACE1BACE2RENOPRD1
SCHEMBL7413268 0.88 GNPAT (0.47) CASP1BACE1BACE2ACE
SCHEMBL7425546 0.84 CASP1 (0.54) CASP1BACE1BACE2RENOPRD1
SCHEMBL5081623 0.84 CASP1 (0.60) CASP1BACE1BACE2RENOPRD1
SCHEMBL7410461 0.83 CASP3 (0.46) CASP1BACE1BACE2CASP3CASP7
SCHEMBL7285000 0.82 CASP1 (0.64) CASP1BACE1BACE2ACEREN
SCHEMBL5686946 0.80 CASP1 (0.55) CASP1BACE1BACE2ACEREN
SCHEMBL17732666 0.80 BACE1 (0.51) CASP1BACE1BACE2ACEREN
SCHEMBL17732682 0.80 GNPAT (0.60) BACE1ACEREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014777-A1 PEPTIDYL DERIVATIVES AS INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME MERCK & CO., INC. (US) 1993-08-05 WO disclosed