SCHEMBL7425673

SCHEMBL7425673

CCCOC(=O)C1=C(C)NC(CF)=C(C(=O)OC)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.68
CACNA1C Q13936 5/20 0.68
OPRM1 P35372 4/20 0.68
KCNH2 Q12809 4/20 0.68
ABCB11 O95342 3/20 0.68
HTR2B P41595 3/20 0.68
SCN5A Q14524 3/20 0.68
CACNA1F O60840 3/20 0.68
CACNA1D Q01668 3/20 0.68
CACNA1S Q13698 3/20 0.68
DRD1 P21728 3/20 0.68
ABCC4 O15439 2/20 0.68
LMNA P02545 2/20 0.68
CYP1A2 P05177 2/20 0.68
ADORA2A P29274 2/20 0.68
ADORA1 P30542 2/20 0.68
SCN1A P35498 2/20 0.68
SCN2A Q99250 2/20 0.68
SCN3A Q9NY46 2/20 0.68
CACNA1B Q00975 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434487 0.93 CYP1A2 (0.57) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL7158381 0.92 ADORA3 (0.80) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL7438852 0.91 CYP1A2 (0.55) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL7434261 0.91 CYP2C9 (0.55) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL6727785 0.88 CACNA1D (0.72) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL10909420 0.86 ADORA3 (0.77) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL7431523 0.86 TBXA2R (0.54) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL7425671 0.85 CYP1A2 (0.69) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL7430547 0.85 TBXA2R (0.56) ADORA3CACNA1COPRM1KCNH2ABCB11
SCHEMBL11824944 0.85 CYP1A2 (0.82) ADORA3CACNA1COPRM1KCNH2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP claimed
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP disclosed