SCHEMBL7158381

SCHEMBL7158381

CCCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.80
CYP1A2 P05177 4/20 0.80
HIF1A Q16665 4/20 0.80
CACNA1C Q13936 3/20 0.80
LMNA P02545 3/20 0.80
CYP3A4 P08684 3/20 0.80
MAPT P10636 3/20 0.80
CYP2C9 P11712 3/20 0.80
CYP2C19 P33261 3/20 0.80
KMT2A Q03164 3/20 0.80
ABCC4 O15439 2/20 0.80
CACNA1F O60840 2/20 0.80
ABCB11 O95342 2/20 0.80
ADORA2A P29274 2/20 0.80
ADORA1 P30542 2/20 0.80
OPRM1 P35372 2/20 0.80
SCN1A P35498 2/20 0.80
HTR2B P41595 2/20 0.80
CACNA1D Q01668 2/20 0.80
KCNH2 Q12809 2/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6727785 0.96 CACNA1D (0.72) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL10909420 0.94 ADORA3 (0.77) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL11824944 0.92 CYP1A2 (0.82) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL5085498 0.92 ADORA3 (0.86) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL7425673 0.92 ADORA3 (0.68) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL10899662 0.92 CACNA1C (0.74) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL10901029 0.92 CACNA1C (0.74) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL6727797 0.91 CACNA1B (0.70) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL9673129 0.91 ADORA3 (0.80) ADORA3CYP1A2HIF1ACACNA1CLMNA
SCHEMBL9175041 0.91 ADORA3 (0.80) ADORA3CYP1A2HIF1ACACNA1CLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545028-B2 Antiepileptic agents, hypotensive agents; monitoring membrane potentials NEUROSEARCH A/S (DK) 2003-04-08 US claimed
US-20020119989-A1 Chemical compounds having ion channel blocking activity for the treatment of immune dysfunction ANIONA APS (DK) 2002-08-29 US claimed
US-6545028-B2 Antiepileptic agents, hypotensive agents; monitoring membrane potentials NEUROSEARCH A/S (DK) 2003-04-08 US disclosed
US-20020119989-A1 Chemical compounds having ion channel blocking activity for the treatment of immune dysfunction ANIONA APS (DK) 2002-08-29 US disclosed
US-3932645-A CORONARY VASODILATORS, HYPOTENSIVE AGENTS FARBENFABRIKEN BAYER AG (DT) 1976-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020119989-A1 Chemical compounds having ion channel blocking activity for the treatment of immune dysfunction KCNN2, KCNN1, KCNJ2 ADORA3 1409/4885CYP1A2 3170/4885HIF1A 2396/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.