SCHEMBL7425870

SCHEMBL7425870

COc1cc(CC(=O)NC2CCN(Cc3ccccc3)CC2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.72

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 14/20 0.72
TSHR P16473 1/20 0.62
ALDH1A1 P00352 1/20 0.57
CCR8 P51685 1/20 0.57
KDM4E B2RXH2 1/20 0.56
HSD17B10 Q99714 1/20 0.56
ITGB1 P05556 1/20 0.56
ITGA4 P13612 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7387042 0.91 ITGB1 (0.67) SIGMAR1TSHRALDH1A1ITGB1ITGA4
SCHEMBL7424843 0.89 SIGMAR1 (0.57) SIGMAR1TSHRITGB1ITGA4
SCHEMBL7430374 0.85 ITGA4 (0.64) SIGMAR1TSHRITGB1ITGA4
SCHEMBL7422099 0.85 ITGA4 (0.55) SIGMAR1TSHRITGB1ITGA4
SCHEMBL7392683 0.84 ITGA4 (0.57) SIGMAR1ALDH1A1KDM4EITGB1ITGA4
SCHEMBL7423342 0.82 ITGA4 (0.62) SIGMAR1ITGB1ITGA4
SCHEMBL7431406 0.80 ITGA4 (0.63) SIGMAR1TSHRITGB1ITGA4
SCHEMBL7425032 0.80 ITGA4 (0.64) SIGMAR1TSHRITGB1ITGA4
SCHEMBL4683165 0.79 ITGA4 (0.67) TSHRALDH1A1ITGB1ITGA4
SCHEMBL7425429 0.79 ITGA4 (0.56) SIGMAR1ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed