SCHEMBL7425958

SCHEMBL7425958

Nc1nccc2ccc(CN(CC(=O)N3CCCCC3)C(=O)O)cc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ECE2 P0DPD6 1/20 0.37
KLKB1 P03952 6/20 0.37
F10 P00742 3/20 0.36
PRMT3 O60678 2/20 0.36
ROCK1 Q13464 2/20 0.35
KLK1 P06870 4/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35
F2 P00734 2/20 0.35
PRSS1 P07477 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
RAB9A P51151 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MAP4K1 Q92918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431443 0.82 KLKB1 (0.44) KLKB1ROCK1KLK1MAP4K1
SCHEMBL15955605 0.74 NPC1 (0.55) HDAC1HDAC6HPGDRAB9A
SCHEMBL7702471 0.73 F2 (0.42) KLKB1F10KLK1HPGDF2
SCHEMBL1189517 0.73 NPC1 (0.57) HDAC1HDAC6RAB9A
SCHEMBL6439089 0.72 F2 (0.50) KLKB1F10F2PRSS1
SCHEMBL27201339 0.70 RAB9A (0.52) KLKB1KLK1HPGDRAB9A
SCHEMBL30885298 0.70 RAB9A (0.52) KLKB1KLK1HPGDRAB9A
SCHEMBL6983681 0.67 F2 (0.42) F10HPGDF2
SCHEMBL6983215 0.66 PLAU (0.60) KLKB1ROCK1PRSS1
SCHEMBL6982094 0.66 ROCK1 (0.53) KLKB1ROCK1PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975600-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS Akzo Nobel N.V. (NL) 2000-02-02 EP disclosed
WO-1998047876-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS AKZO NOBEL N.V. (NL) 1998-10-29 WO disclosed