SCHEMBL7426977

SCHEMBL7426977

CN(C#N)C(=O)C1(NC(=O)c2ccc(-c3csc(N4CCOCC4)n3)cc2)CCCCC1

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSB P07858 17/20 0.74
CTSS P25774 17/20 0.74
CTSL P07711 16/20 0.74
CTSK P43235 5/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6183543 0.85 CTSB (1.00) CTSBCTSSCTSLCTSK
SCHEMBL6185943 0.83 CTSB (0.68) CTSBCTSSCTSLCTSK
SCHEMBL1838437 0.80 CTSB (0.67) CTSBCTSSCTSLCTSK
SCHEMBL6182540 0.80 CTSB (0.52) CTSBCTSSCTSLCTSK
SCHEMBL1842461 0.80 CTSB (0.66) CTSBCTSSCTSLCTSK
SCHEMBL6181475 0.79 CTSB (0.73) CTSBCTSSCTSLCTSK
SCHEMBL6180697 0.78 CTSL (0.60) CTSBCTSSCTSLCTSK
SCHEMBL13798777 0.77 CTSB (0.76) CTSBCTSSCTSLCTSK
SCHEMBL13798776 0.77 CTSB (0.76) CTSBCTSSCTSLCTSK
SCHEMBL12661358 0.77 CTSB (0.75) CTSBCTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO disclosed