SCHEMBL7427282

SCHEMBL7427282

CC[C@H](C)[C@H](NC(=O)Cc1ccccn1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.48
NFE2L2 Q16236 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
POLB P06746 2/20 0.48
PTPRA P18433 1/20 0.44
ADAMTS4 O75173 1/20 0.43
ALDH1A1 P00352 2/20 0.43
FPR2 P25090 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ATM Q13315 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PSMB5 P28074 1/20 0.42
ANPEP P15144 1/20 0.41
CA2 P00918 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301586 0.83 POLB (0.60) CYP2C9CYP2C19POLBALDH1A1KMT2A
SCHEMBL7387341 0.83 POLB (0.60) CYP2C9CYP2C19POLBALDH1A1KMT2A
SCHEMBL7438190 0.81 POLB (0.41) KEAP1NFE2L2CYP2C19POLBALDH1A1
SCHEMBL7310554 0.81 RAB9A (0.55) CYP2C9CYP2C19POLBADAMTS4MEN1
SCHEMBL7310548 0.81 RAB9A (0.55) CYP2C9CYP2C19POLBADAMTS4MEN1
SCHEMBL9830901 0.80 POLB (0.59) CYP2C9CYP2C19POLBALDH1A1MEN1
SCHEMBL5917035 0.80 POLB (0.59) CYP2C9CYP2C19POLBALDH1A1MEN1
SCHEMBL5917036 0.80 POLB (0.59) CYP2C9CYP2C19POLBALDH1A1MEN1
SCHEMBL16114864 0.80 POLB (0.59) CYP2C9CYP2C19POLBALDH1A1MEN1
SCHEMBL7393135 0.80 CA2 (0.60) KEAP1NFE2L2CYP2C9CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665215-A1 1,4-Diamino-2,3-dihydroxybutanes THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-08-02 EP disclosed
US-5430155-A Viricides, treatment of AIDS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-07-04 US disclosed
US-5294720-A Viricides THE DUPONT MERCK PHARMACEUTICAL CO. (US) 1994-03-15 US disclosed
EP-0532693-A1 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-03-24 EP disclosed
WO-1991018866-A2 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-12 WO disclosed