SCHEMBL7427342

SCHEMBL7427342

CC(CCNC(=N)N)NS(=O)(=O)c1cccc2cnccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCG P05129 4/20 0.56
PRKCZ Q05513 4/20 0.56
PRKCD Q05655 4/20 0.56
PRKD3 O94806 3/20 0.56
PRKCB P05771 3/20 0.56
PRKCA P17252 3/20 0.56
PRKCH P24723 3/20 0.56
PRKCI P41743 3/20 0.56
PRKCE Q02156 3/20 0.56
PRKCQ Q04759 3/20 0.56
PRKD1 Q15139 3/20 0.56
CYP3A4 P08684 3/20 0.56
CYP2D6 P10635 3/20 0.56
NFKB1 P19838 3/20 0.56
PRKACA P17612 3/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
PRKACG P22612 2/20 0.56
PRKACB P22694 2/20 0.56
TP53 P04637 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423209 0.89 PRKD3 (0.52) PRKCGPRKCZPRKCDPRKD3PRKCB
SCHEMBL2903275 0.88 PRKD3 (0.51) PRKCGPRKCZPRKCDPRKD3PRKCB
SCHEMBL1272417 0.87 PRKACA (0.70) PRKCGPRKCZPRKCDPRKD3PRKCB
Hydrochloric Acid SCHEMBL1165287 0.86 LMNA (0.70) PRKCGPRKCZPRKCDPRKD3PRKCB
Hydrochloric Acid SCHEMBL30084456 0.86 LMNA (0.70) PRKCGPRKCZPRKCDPRKD3PRKCB
Hydrochloric Acid SCHEMBL5177180 0.86 LMNA (0.70) PRKCGPRKCZPRKCDPRKD3PRKCB
SCHEMBL7431555 0.85 MELK (0.54) PRKCGPRKCZPRKCDPRKD3PRKCB
SCHEMBL7427348 0.85 PRKACA (0.64) PRKCGPRKCZPRKCDPRKD3PRKCB
SCHEMBL7430584 0.85 PRKCG (0.50) PRKCGPRKCZPRKCDPRKD3PRKCB
SCHEMBL7434254 0.84 PRKACA (0.59) PRKCGPRKCZPRKCDPRKD3PRKCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4709032-A VASODILATION AND HYPOTENSIVE AGENT ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1987-11-24 US disclosed
US-4634770-A VASODILATORS, HYPOTENSIVES ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1987-01-06 US disclosed
EP-0109023-A1 Isoquinolinesulfonamide derivatives and process for the preparation thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1984-05-23 EP disclosed