SCHEMBL7427699

SCHEMBL7427699

CCCOC(=O)C1=C(C)NC(CF)=C(C(=O)OC)C1c1cc([N+](=O)[O-])ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.52
CACNA1C Q13936 4/20 0.51
HIF1A Q16665 3/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
MAPT P10636 3/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.51
GPR55 Q9Y2T6 1/20 0.51
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51
THPO P40225 1/20 0.51
HTR1A P08908 2/20 0.49
ADRA2A P08913 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430466 0.91 ADORA3 (0.53) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL7426393 0.86 ADORA3 (0.54) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL11829575 0.86 ADORA3 (0.69) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL11376477 0.83 CACNA1C (0.56) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL11690943 0.82 ADORA3 (0.61) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL7434261 0.82 CYP2C9 (0.55) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL7425673 0.81 ADORA3 (0.68) ADORA3CACNA1CHIF1AKMT2AMAPT
SCHEMBL7273495 0.80 CYP1A2 (0.65) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL7273500 0.80 CYP1A2 (0.65) ADORA3CACNA1CHIF1AMEN1KMT2A
SCHEMBL7434487 0.80 CYP1A2 (0.57) ADORA3CACNA1CHIF1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP claimed