SCHEMBL7427967

SCHEMBL7427967

CC(C)CC(N)C(=O)NC1CCCN(S(=O)(=O)c2ccccc2)C[C@@H]1O

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 6/20 0.53
LARS1 Q9P2J5 2/20 0.47
CYP2C19 P33261 1/20 0.46
MMP2 P08253 1/20 0.45
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5098782 1.00 CACNA1B (0.53) CACNA1BLARS1CYP2C19MMP2LMNA
SCHEMBL5105401 0.90 CACNA1B (0.47) CACNA1BMMP2LMNAALDH1A1
SCHEMBL5092886 0.89 CACNA1B (0.57) CACNA1BLARS1LMNAALDH1A1
SCHEMBL5105633 0.89 ALDH1A1 (0.49) CACNA1BLMNASMN1; SMN2ALDH1A1
SCHEMBL7427831 0.88 CACNA1B (0.53) CACNA1BLMNAALDH1A1
SCHEMBL4686499 0.86 CTSK (0.49) CACNA1B
SCHEMBL5971807 0.86 CTSK (0.49) CACNA1B
SCHEMBL14131846 0.85 CACNA1B (0.42) CACNA1BLARS1MMP2
SCHEMBL5096704 0.85 CACNA1B (0.42) CACNA1BLARS1MMP2
SCHEMBL5105253 0.83 CACNA1B (0.45) CACNA1BLARS1LMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed