SCHEMBL7428131

SCHEMBL7428131

CC(C)(C)OC(=O)NCCCC(CN)Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
GAA P10253 1/20 0.53
KMT2A Q03164 1/20 0.53
IDO1 P14902 1/20 0.48
CTSK P43235 4/20 0.47
CTSS P25774 3/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
PAX8 Q06710 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ATM Q13315 1/20 0.46
MMP1 P03956 1/20 0.46
MMP3 P08254 1/20 0.46
MMP9 P14780 1/20 0.46
MAPT P10636 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
AKT1 P31749 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12295159 0.85 ATM (0.53) IDO1CTSKCTSSCTSLCTSB
SCHEMBL18748463 0.85 ATM (0.53) IDO1CTSKCTSSCTSLCTSB
SCHEMBL24003388 0.84 MEN1 (0.69) MEN1GAAKMT2AIDO1CTSK
SCHEMBL9074865 0.84 MEN1 (0.69) MEN1GAAKMT2AIDO1CTSK
SCHEMBL3722339 0.84 MEN1 (0.57) MEN1GAAKMT2AIDO1CTSK
SCHEMBL6335082 0.84 MEN1 (0.57) MEN1GAAKMT2AIDO1CTSK
SCHEMBL7427102 0.83 SYK (0.49) IDO1CTSKCTSSCTSLCTSB
SCHEMBL15159959 0.81 ATM (0.62) MEN1GAAKMT2ACTSKCTSS
SCHEMBL12452003 0.80 IDO1 (0.52) MEN1GAAKMT2AIDO1CTSK
SCHEMBL14598335 0.79 CTSS (0.51) MEN1GAAKMT2AIDO1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4709032-A VASODILATION AND HYPOTENSIVE AGENT ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1987-11-24 US disclosed
US-4634770-A VASODILATORS, HYPOTENSIVES ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1987-01-06 US disclosed
EP-0109023-A1 Isoquinolinesulfonamide derivatives and process for the preparation thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1984-05-23 EP disclosed