SCHEMBL7428579

SCHEMBL7428579

COc1ccccc1COc1ccc(CC(=O)N2CCCC2c2cc(CCC(=O)O)on2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 7/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
YAP1 P46937 1/20 0.41
SCD5 Q86SK9 2/20 0.40
SCD O00767 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CPT1A P50416 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
PPARD Q03181 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484778 0.92 FFAR1 (0.45) FFAR1NPC1RAB9ACPT1AFFAR4
SCHEMBL7488757 0.89 FFAR1 (0.42) FFAR1NPC1RAB9ACPT1AFFAR4
SCHEMBL7481567 0.89 FFAR1 (0.45) FFAR1NPC1RAB9AYAP1FFAR4
SCHEMBL7424997 0.87 FFAR1 (0.52) FFAR1NPC1RAB9ASCD5CPT1A
SCHEMBL7427523 0.87 NPC1 (0.49) FFAR1NPC1RAB9ASCD5SCD
SCHEMBL7434473 0.87 NPC1 (0.45) FFAR1NPC1RAB9ASCD5SCD
SCHEMBL7433472 0.86 CPT1A (0.42) FFAR1YAP1CPT1AFFAR4
SCHEMBL7487553 0.86 FFAR1 (0.42) FFAR1NPC1RAB9ACPT1AFFAR4
SCHEMBL7433078 0.86 FFAR1 (0.42) FFAR1NPC1RAB9ACPT1AFFAR4
SCHEMBL7429711 0.85 FFAR4 (0.42) FFAR1SCD5SCDFFAR4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244656-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES Pfizer Products Inc. (US) 2002-10-02 EP disclosed
WO-2001051487-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PRODUCTS INC. (US) 2001-07-19 WO disclosed