SCHEMBL7424997

SCHEMBL7424997

N#Cc1ccccc1COc1ccc(CC(=O)N2CCCC2c2cc(CCC(=O)O)on2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 5/20 0.52
MAOB P27338 1/20 0.41
AKR1B1 P15121 1/20 0.40
CPT1A P50416 5/20 0.39
CPT2 P23786 3/20 0.39
SCD5 Q86SK9 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KCNH2 Q12809 1/20 0.37
GYS1 P13807 1/20 0.37
FFAR4 Q5NUL3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484778 0.89 FFAR1 (0.45) FFAR1CPT1ANPC1RAB9AFFAR4
SCHEMBL7488757 0.89 FFAR1 (0.42) FFAR1MAOBCPT1ANPC1RAB9A
SCHEMBL7481567 0.88 FFAR1 (0.45) FFAR1NPC1RAB9AFFAR4
SCHEMBL7428579 0.87 FFAR1 (0.43) FFAR1CPT1ASCD5NPC1RAB9A
SCHEMBL7434473 0.85 NPC1 (0.45) FFAR1MAOBCPT1ACPT2SCD5
SCHEMBL7433472 0.84 CPT1A (0.42) FFAR1CPT1AFFAR4
SCHEMBL7487553 0.84 FFAR1 (0.42) FFAR1CPT1ANPC1RAB9AFFAR4
SCHEMBL7433078 0.84 FFAR1 (0.42) FFAR1CPT1ANPC1RAB9AFFAR4
SCHEMBL7435979 0.84 CPT1A (0.43) FFAR1CPT1ANPC1RAB9AFFAR4
SCHEMBL7542862 0.84 CPT1A (0.42) FFAR1MAOBCPT1ACPT2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244656-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES Pfizer Products Inc. (US) 2002-10-02 EP disclosed
WO-2001051487-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PRODUCTS INC. (US) 2001-07-19 WO disclosed