SCHEMBL7428665

SCHEMBL7428665

CC(C)(C)[Si](C)(C)Oc1ccc(C=O)c(N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.46
CA1 P00915 4/20 0.46
CA9 Q16790 4/20 0.46
PREP P48147 4/20 0.38
ALDH1A1 P00352 2/20 0.37
ERN1 O75460 1/20 0.36
TRIM24 O15164 1/20 0.36
TYR P14679 1/20 0.36
TRIM33 Q9UPN9 1/20 0.36
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
TUBB1 Q9H4B7 2/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1070012 0.84 CA12 (0.48) CA12CA1CA9PREPALDH1A1
SCHEMBL14240879 0.84 CA12 (0.48) CA12CA1CA9PREPALDH1A1
SCHEMBL22078670 0.83 CA12 (0.47) CA12CA1CA9PREPALDH1A1
SCHEMBL19810818 0.83 ALDH1A1 (0.49) CA12CA1CA9PREPALDH1A1
SCHEMBL17494765 0.81 CA12 (0.46) CA12CA1CA9PREPALDH1A1
SCHEMBL7618394 0.81 TYR (0.58) CA12CA1CA9PREPALDH1A1
SCHEMBL2511093 0.81 CA12 (0.46) CA12CA1CA9PREPALDH1A1
SCHEMBL6841139 0.81 CA12 (0.48) CA12CA1CA9PREPALDH1A1
SCHEMBL2199657 0.81 CA12 (0.48) CA12CA1CA9PREPALDH1A1
SCHEMBL5383976 0.80 ALDH1A1 (0.63) CA12CA1CA9ALDH1A1ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107954-A1 2-OXO-$i(2H)-QUINOLINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-06-20 EP disclosed
WO-2000012479-A1 2-OXO-2H-QUINOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-03-09 WO disclosed