SCHEMBL7428865

SCHEMBL7428865

[c]1ccc2c3c(ccc2c1)OCO3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 4/20 0.38
MAPT P10636 4/20 0.38
HPGD P15428 4/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
MAPK1 P28482 3/20 0.38
MEN1 O00255 3/20 0.38
LMNA P02545 3/20 0.38
KMT2A Q03164 3/20 0.38
HSD17B10 Q99714 3/20 0.38
ACHE P22303 3/20 0.38
CYP1A2 P05177 3/20 0.38
RGS17 Q9UGC6 2/20 0.38
BAD Q92934 2/20 0.38
RGS12 O14924 2/20 0.38
TP53 P04637 2/20 0.38
CYP3A4 P08684 2/20 0.38
ALOX15 P16050 2/20 0.38
ALOX12 P18054 2/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431153 0.86 ALDH1A1 (0.38) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL403982 0.73 BAD (0.49) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL30400843 0.73 BAD (0.49) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL70608 0.71 ALDH1A1 (0.33) ALDH1A1HSD17B10TSHRTDP1
SCHEMBL7537851 0.70 KDM4E (0.33) KDM4EMAPTHPGDMEN1KMT2A
SCHEMBL3142725 0.69 CYP3A4 (0.38) ALDH1A1MAPK1HSD17B10CYP3A4TDP1
SCHEMBL7533311 0.68 MTNR1A (0.34) KDM4EHPGDHSD17B10ACHECYP1A2
SCHEMBL3971384 0.68 KDM4E (0.43) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL20662 0.68
SCHEMBL2282037 0.67 HPRT1 (0.39) ALDH1A1HSD17B10TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283310-B1 N-BENZHYDRYL-SUBSTITUTED HETEROCYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE Sankyo Company Limited (JP) 1993-05-26 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
US-5028610-A Calcium Channel Blockers SANKYO COMPANY LIMITED (JP) 1991-07-02 US disclosed
EP-0283310-A1 N-Benzhydryl-substituted heterocyclic derivatives, their preparation and their use Sankyo Company Limited (JP) 1988-09-21 EP disclosed