SCHEMBL7428878

SCHEMBL7428878

C[C@@H](CC(N)=O)CC(=O)NC1CCCN(C(=O)Cc2cccc(-c3ccccn3)c2)CC1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.53
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41
CTSS P25774 2/20 0.41
POLB P06746 2/20 0.38
MAP3K12 Q12852 1/20 0.37
KDM6B O15054 1/20 0.36
KDM5C P41229 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
KDM3A Q9Y4C1 1/20 0.36
TP53BP1 Q12888 1/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 1/20 0.35
PDE2A O00408 1/20 0.35
LCK P06239 1/20 0.35
BTK Q06187 1/20 0.34
LMNA P02545 1/20 0.34
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691184 0.88 CTSK (0.53) CTSKCTSLCTSBCTSSPOLB
SCHEMBL6404534 0.84 CTSK (0.64) CTSKCTSLCTSBCTSSPOLB
SCHEMBL5098711 0.84 CTSK (0.64) CTSKCTSLCTSBCTSSPOLB
SCHEMBL6578142 0.84 CTSK (0.48) CTSKCTSLCTSBCTSSPOLB
SCHEMBL5098703 0.84 CTSK (0.52) CTSKCTSLCTSBCTSSPOLB
SCHEMBL7429714 0.82 CTSK (0.64) CTSKCTSLCTSBCTSSPOLB
SCHEMBL5105817 0.79 CTSK (0.49) CTSKCTSLCTSBCTSSPOLB
SCHEMBL4689761 0.78 CTSK (0.63) CTSKCTSLCTSBCTSS
SCHEMBL7037376 0.78 CTSK (0.63) CTSKCTSLCTSBCTSS
SCHEMBL4689758 0.78 CTSK (0.63) CTSKCTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed