SCHEMBL7429686

SCHEMBL7429686

CC(=O)SCC(Cc1cccnc1)C(=O)Nc1cccc(C(=O)OCc2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.55
CYP3A4 P08684 4/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ABCC3 O15438 1/20 0.50
NR1I2 O75469 1/20 0.50
ABCB11 O95342 1/20 0.50
NR3C1 P04150 1/20 0.50
RARG P13631 1/20 0.50
CNR1 P21554 1/20 0.50
OPRK1 P41145 1/20 0.50
NR1H2 P55055 1/20 0.50
PPARA Q07869 1/20 0.50
NR1H3 Q13133 1/20 0.50
NR1I3 Q14994 1/20 0.50
LMNA P02545 1/20 0.49
KMT2A Q03164 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7433987 0.96 RAB9A (0.52) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7432730 0.91 RAB9A (0.64) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7431935 0.88 TSHR (0.50) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9456817 0.86 TSHR (0.42) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL7438031 0.86 RAB9A (0.57) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7436824 0.85 RAB9A (0.56) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL7429379 0.84 RAB9A (0.55) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7433382 0.83 MAPT (0.56) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL7428252 0.83 RAB9A (0.52) RAB9ACYP3A4LMNAKMT2ATDP1
SCHEMBL7430654 0.82 RAB9A (0.50) RAB9ACYP3A4CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210266-A Analgesic enkephalinase inhibitors DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5179125-A Analgesics DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-01-12 US disclosed
EP-0318859-A2 N-substituted mercaptopropanamide derivatives Dainippon Pharmaceutical Co., Ltd. (JP) 1989-06-07 EP disclosed