SCHEMBL7430368

SCHEMBL7430368

Nc1cc(N2CCCCC2)cc2nc(-c3ccco3)nn12

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.66
ADORA1 P30542 3/20 0.56
ALDH1A1 P00352 1/20 0.52
ADORA3 P0DMS8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480538 0.99 ADORA2A (0.65) ADORA2AADORA1ALDH1A1
SCHEMBL7482833 0.88 ADORA2A (0.56) ADORA2AADORA1ADORA3
SCHEMBL6622137 0.81 ADORA2A (0.68) ADORA2AADORA1
SCHEMBL7705992 0.80 HPGD (0.45) ADORA2AALDH1A1ADORA3
SCHEMBL6863438 0.80 ADORA2A (1.00) ADORA2AADORA1ALDH1A1
SCHEMBL7709059 0.79 SMN1; SMN2 (0.45) ADORA2AALDH1A1ADORA3
SCHEMBL6870294 0.78 ADORA2A (1.00) ADORA2AADORA1ALDH1A1
SCHEMBL7427470 0.77 ADORA2A (0.59) ADORA2AADORA1
SCHEMBL7711835 0.76 ADORA2A (0.64) ADORA2A
SCHEMBL7703248 0.76 ADORA2A (0.46) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP claimed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO claimed
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed