SCHEMBL7703248

SCHEMBL7703248

Nc1cc(N2CCc3c([nH]c4ccccc34)C2)cc2nc(-c3ccco3)nn12

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.46
DHFR P00374 1/20 0.39
GBA1 P04062 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705975 0.86 GBA1 (0.48) DHFRGBA1KDM4E
SCHEMBL7480538 0.77 ADORA2A (0.65) ADORA2AADORA1
SCHEMBL7430368 0.76 ADORA2A (0.66) ADORA2AADORA1
SCHEMBL7482833 0.74 ADORA2A (0.56) ADORA2AADORA1
SCHEMBL6632327 0.73 ADRA2A (0.59) ADORA2ADHFR
SCHEMBL6867881 0.70 ADORA2A (0.63) ADORA2A
SCHEMBL7427470 0.66 ADORA2A (0.59) ADORA2AADORA1
SCHEMBL21588453 0.66 KDM4E (0.51) DHFRKDM4E
SCHEMBL21588421 0.66 DHFR (0.53) DHFRGBA1KDM4E
SCHEMBL7711605 0.66 ADORA2A (0.55) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed