SCHEMBL7430619

SCHEMBL7430619

NC(Cc1cn(S(=O)(=O)c2ccccc2)c2ccc(OCc3ccccc3)cc12)OC(=O)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 15/20 0.60
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR1E P28566 1/20 0.45
HTR1F P30939 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 1/20 0.44
PPARG P37231 2/20 0.43
PPARD Q03181 2/20 0.43
PPARA Q07869 2/20 0.43
MEN1 O00255 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
LTA4H P09960 1/20 0.41
PLA2G2A P14555 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433712 0.83 HTR6 (0.58) HTR6HTR1ADRD2HTR1DHTR1B
Oxalic Acid SCHEMBL7430614 0.82 HTR6 (0.71) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7436733 0.81 HTR6 (0.57) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL12344906 0.76 HTR6 (0.64) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL5030681 0.75 HTR6 (0.66) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL5505546 0.75 HTR6 (1.00) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7441788 0.75 HTR6 (0.61) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL2882506 0.74 MEN1 (0.65) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7433688 0.74 HTR6 (0.58) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL2886894 0.73 HTR6 (0.63) HTR6HTR1ADRD2HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187805-B1 TREATING CONDITION FOR WHICH SELECTIVE AGONISM OR ANTAGONISM OF 5-HT-6 RECEPTORS IS INDICATED BY ADMINISTERING COMPOUNDS SUCH AS N,N-DIMETHYL 2-(1-(BENZENESULPHONYL)-5-METHOXY-1H-INDOL-3-YL)ETHYLAMINE MERCK SHARP & DOHME LTD. (GB) 2001-02-13 US disclosed