SCHEMBL7436733

SCHEMBL7436733

N#Cc1ccc2c(c1)c(CC(N)OC(=O)C(=O)O)cn2S(=O)(=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 18/20 0.57
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR1E P28566 1/20 0.40
HTR1F P30939 1/20 0.40
HTR7 P34969 1/20 0.40
DRD3 P35462 1/20 0.40
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
IDE P14735 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433712 0.85 HTR6 (0.58) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7430619 0.81 HTR6 (0.60) HTR6HTR1ADRD2HTR1DHTR1B
Oxalic Acid SCHEMBL7436726 0.80 HTR6 (0.69) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL5500213 0.78 HTR6 (0.74) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7433688 0.75 HTR6 (0.58) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7441106 0.73 HTR6 (0.48) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL5512690 0.73 HTR6 (1.00) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL27867109 0.73 HTR6 (0.70) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL28073957 0.73 HTR6 (0.70) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL7441788 0.71 HTR6 (0.61) HTR6HTR1ADRD2HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187805-B1 TREATING CONDITION FOR WHICH SELECTIVE AGONISM OR ANTAGONISM OF 5-HT-6 RECEPTORS IS INDICATED BY ADMINISTERING COMPOUNDS SUCH AS N,N-DIMETHYL 2-(1-(BENZENESULPHONYL)-5-METHOXY-1H-INDOL-3-YL)ETHYLAMINE MERCK SHARP & DOHME LTD. (GB) 2001-02-13 US disclosed