SCHEMBL7430711

SCHEMBL7430711

[c]1ccc(-c2ccncc2-c2nnn[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 6/20 0.39
CYP1A2 P05177 2/20 0.30
CYP2D6 P10635 2/20 0.30
CYP2A6 P11509 2/20 0.30
CYP2B6 P20813 2/20 0.30
CYP2C19 P33261 2/20 0.30
CYP2E1 P05181 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435406 0.95 RPS6KA3 (0.38) RPS6KA3
SCHEMBL4712959 0.82 DCUN1D1 (0.36)
SCHEMBL6176 0.77
SCHEMBL7446017 0.76 ESR1 (0.32)
SCHEMBL7429132 0.76 ESR1 (0.32)
SCHEMBL27513088 0.74
SCHEMBL7256207 0.73 TDO2 (0.37) CYP1A2CYP2D6CYP2A6CYP2B6CYP2C19
SCHEMBL28594934 0.73 RPS6KA3 (0.54) RPS6KA3CYP1A2CYP2D6CYP2A6CYP2B6
SCHEMBL28596691 0.73 RPS6KA3 (0.54) RPS6KA3CYP1A2CYP2D6CYP2A6CYP2B6
SCHEMBL7431528 0.73 MEN1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed