SCHEMBL7430862

SCHEMBL7430862

CN([C@@]1(Cc2cccc(C#N)c2)CCNC1=O)S(=O)(=O)c1ccc(-c2ccnc([S+](C)[O-])n2)s1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8623715 0.76 F10 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7418409 0.72 F10 (0.58)
SCHEMBL7426894 0.69 F10 (0.44) ALDH1A1MAPT
SCHEMBL7425777 0.64 GABRA1 (0.37) MAPT
SCHEMBL8626510 0.63 F10 (0.43)
SCHEMBL7429862 0.59 HRH3 (0.41)
SCHEMBL4493324 0.56 MAPT (0.36) ALDH1A1MAPT
SCHEMBL7423776 0.56 EPHX1 (0.41)
SCHEMBL12423089 0.56 IKBKB (0.60)
SCHEMBL3819160 0.56 CYP3A4 (0.39) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894088-A4 SUBSTITUTED SULFONIC ACID N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2001-12-05 EP disclosed
EP-0894088-A1 SUBSTITUTED SULFONIC ACID N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-02-03 EP disclosed
WO-1998024784-A1 SUBSTITUTED SULFONIC ACID N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-06-11 WO disclosed