SCHEMBL7430896

SCHEMBL7430896

O=C(Cl)c1cccnc1-c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.53
KDM4E B2RXH2 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 1/20 0.45
PTGS2 P35354 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MKNK1 Q9BUB5 5/20 0.44
MKNK2 Q9HBH9 4/20 0.44
RORB Q92753 1/20 0.43
KMO O15229 2/20 0.42
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
POLB P06746 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PIM1 P11309 1/20 0.41
KCNN4 O15554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5145882 0.85 KDM4E (0.67) CYP2A6KDM4ETDP1ALDH1A1CYP1A2
SCHEMBL29575496 0.83 MKNK1 (0.55) CYP2A6KDM4ETDP1MKNK1MKNK2
Hydrochloric Acid SCHEMBL22719435 0.83 KDM4E (0.65) CYP2A6KDM4ETDP1ALDH1A1CYP1A2
SCHEMBL1571384 0.83 MKNK1 (0.55) CYP2A6KDM4ETDP1MKNK1MKNK2
SCHEMBL3263627 0.82 KDM4E (0.65) KDM4ETDP1ALDH1A1CYP3A4L3MBTL1
Nitrous Acid SCHEMBL28224285 0.80 KDM4E (0.59) CYP2A6KDM4ETDP1ALDH1A1CYP3A4
SCHEMBL38658131 0.76 RAB9A (0.60) CYP2A6KDM4EALDH1A1MKNK1MKNK2
SCHEMBL7430892 0.76 CYP2A6 (0.48) CYP2A6KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL31635952 0.74 PTGS2 (0.64) CYP2A6KDM4ETDP1ALDH1A1CYP1A2
SCHEMBL30032 0.74 PTGS2 (0.64) CYP2A6KDM4ETDP1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183239-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2002-03-06 EP disclosed
WO-2000069821-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2000-11-23 WO disclosed