SCHEMBL7430992

SCHEMBL7430992

COC(=O)Oc1cccc2[nH]cnc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
DRD2 P14416 2/20 0.45
DRD3 P35462 2/20 0.45
DRD4 P21917 1/20 0.45
BRD4 O60885 2/20 0.45
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
FAAH O00519 1/20 0.43
CNR1 P21554 1/20 0.43
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4604974 0.84 PARP1 (0.46) PARP1DRD2DRD3DRD4BRD4
SCHEMBL7432212 0.83 PARP1 (0.53) PARP1DRD2DRD3DRD4BRD4
SCHEMBL7519272 0.81 PARP1 (0.59) PARP1DRD2DRD3DRD4BRD4
SCHEMBL25475153 0.79 PARP1 (0.47) PARP1DRD2DRD3DRD4BRD4
SCHEMBL10140 0.79 BRD4 (0.60) PARP1DRD2DRD3DRD4BRD4
SCHEMBL30805278 0.78 PARP1 (0.48) PARP1DRD2DRD3DRD4BRD4
SCHEMBL536589 0.75 PARP1 (0.64) PARP1
Nitric Acid SCHEMBL14695919 0.75 BRD4 (0.50) PARP1DRD2DRD3DRD4BRD4
Nitric Acid SCHEMBL14695921 0.75 BRD4 (0.50) PARP1DRD2DRD3DRD4BRD4
SCHEMBL23123499 0.74 DRD2 (0.46) PARP1DRD2DRD3DRD4BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001051484-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2001-07-19 WO disclosed