SCHEMBL7433281

SCHEMBL7433281

Fc1ccc(C(c2ccncc2)C2CCCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.47
CYP11B2 P19099 1/20 0.47
MAPK14 Q16539 5/20 0.43
MAPK13 O15264 3/20 0.43
MAPK12 P53778 3/20 0.43
MAPK11 Q15759 3/20 0.43
RAF1 P04049 1/20 0.43
MAPK9 P45984 1/20 0.43
MAPKAPK2 P49137 2/20 0.40
DAPK3 O43293 1/20 0.40
ROCK2 O75116 1/20 0.40
CHEK2 O96017 1/20 0.40
PIM1 P11309 1/20 0.40
PLK1 P53350 1/20 0.40
ROCK1 Q13464 1/20 0.40
CDC42BPA Q5VT25 1/20 0.40
AURKB Q96GD4 1/20 0.40
PLK3 Q9H4B4 1/20 0.40
AKT1 P31749 1/20 0.40
GCGR P47871 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257480 0.74 SLC6A3 (0.34)
SCHEMBL18823394 0.74 CYP19A1 (0.49) CYP19A1CYP11B2MAPKAPK2DAPK3ROCK2
SCHEMBL31388237 0.73 PDE4A (0.44) CYP19A1MAPK14PDE4APRCP
SCHEMBL20475315 0.73 SYK (0.38) CYP19A1CYP11B2MAPK14MAPK13MAPK12
SCHEMBL8206213 0.73 SLC6A2 (0.41) NPC1RAB9A
SCHEMBL16269909 0.72 SLC6A2 (0.41)
SCHEMBL29173225 0.71 MAPKAPK2 (0.45) CYP19A1MAPK14MAPK13MAPK12MAPK11
SCHEMBL23882954 0.71 DHODH (0.50) CYP19A1CYP11B2MAPKAPK2DAPK3ROCK2
SCHEMBL8910330 0.71 CYP19A1 (0.41) CYP19A1CYP11B2MAPKAPK2DAPK3ROCK2
SCHEMBL22984539 0.71 DHODH (0.50) CYP19A1CYP11B2MAPKAPK2DAPK3ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed
US-4950674-A Arylalkylheterocyclic amines,N-substituted by aryloxyalkyl group in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-21 US disclosed