SCHEMBL7433345

SCHEMBL7433345

O=C(O)CCCN1Cc2ccccc2C1=O

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.83
ALOX15 P16050 1/20 0.83
TSHR P16473 1/20 0.83
SIRT1 Q96EB6 1/20 0.83
ALDH1A1 P00352 1/20 0.60
HPGD P15428 1/20 0.60
DRD2 P14416 3/20 0.58
DRD5 P21918 3/20 0.58
DRD3 P35462 3/20 0.58
HTR1A P08908 1/20 0.58
HTR7 P34969 2/20 0.56
HDAC3 O15379 1/20 0.56
HDAC4 P56524 1/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC7 Q8WUI4 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC10 Q969S8 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383921 0.94 KDM4E (0.78) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL13593314 0.94 KDM4E (0.78) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL31188916 0.91 KDM4E (1.00) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL315339 0.91 KDM4E (1.00) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL7997184 0.88 KDM4E (0.68) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL11347453 0.84 HDAC3 (0.65) KDM4EALOX15TSHRSIRT1HPGD
SCHEMBL9375738 0.83 KDM4E (0.65) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL7995733 0.82 HDAC6 (0.67) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL30073110 0.82 KDM4E (0.72) KDM4EALOX15TSHRSIRT1ALDH1A1
SCHEMBL30073106 0.82 KDM4E (0.72) KDM4EALOX15TSHRSIRT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375451-A2 Compounds having a renin-inhibiting activity BEECHAM GROUP PLC (GB) 1990-06-27 EP disclosed