SCHEMBL7433470

SCHEMBL7433470

Cc1cc(/C=C/C#N)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.44
UHRF1 Q96T88 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ENPP2 Q13822 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
KCNH2 Q12809 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
DYRK1A Q13627 1/20 0.33
GRM5 P41594 2/20 0.32
AKR1C3 P42330 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ALOX12 P18054 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PDE10A Q9Y233 1/20 0.30
ALOX5 P09917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17053181 1.00 FDPS (0.44) FDPSUHRF1KDM4EENPP2CYP3A4
SCHEMBL7433476 1.00 FDPS (0.44) FDPSUHRF1KDM4EENPP2CYP3A4
SCHEMBL17053184 0.82 DYRK1A (0.49) FDPSUHRF1KDM4ECYP3A4CYP2C9
SCHEMBL7422681 0.78 ENPP2 (0.41) FDPSKDM4EENPP2CYP3A4CYP2C9
SCHEMBL7434021 0.78 ENPP2 (0.41) FDPSKDM4EENPP2CYP3A4CYP2C9
SCHEMBL7422694 0.78 ENPP2 (0.41) FDPSKDM4EENPP2CYP3A4CYP2C9
SCHEMBL7428148 0.77 FDPS (0.44) FDPSKDM4EENPP2CYP3A4CYP2C9
SCHEMBL7428143 0.77 FDPS (0.44) FDPSKDM4EENPP2CYP3A4CYP2C9
SCHEMBL7425838 0.77 FDPS (0.41) FDPSKDM4EENPP2CYP3A4CYP2C9
SCHEMBL7425836 0.77 FDPS (0.41) FDPSKDM4EENPP2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed