SCHEMBL7433498

SCHEMBL7433498

O=C(O)C(Cc1c[nH]cn1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.33
CYP3A4 P08684 1/20 0.33
SLC7A5 Q01650 1/20 0.33
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
LDHA P00338 1/20 0.32
CPB2 Q96IY4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10073663 0.89 PTPRA (0.30) PTPRA
SCHEMBL9555107 0.85 PPARG (0.39) KMT2ALDHACPB2
SCHEMBL9555112 0.85 PPARG (0.39) KMT2ALDHACPB2
SCHEMBL1312464 0.85 PTPRA (0.50) PTPRACYP3A4SLC7A5
SCHEMBL1312465 0.85 PTPRA (0.50) PTPRACYP3A4SLC7A5
SCHEMBL3839517 0.83 PTPRA (0.31) PTPRACYP3A4SLC7A5
Histidine SCHEMBL388563 0.83 SLC7A5 (0.47) CYP3A4SLC7A5KMT2A
SCHEMBL3159235 0.83 APAF1 (0.40) PTPRACYP3A4SLC7A5CPB2
SCHEMBL3670921 0.83 APAF1 (0.40) PTPRACYP3A4SLC7A5CPB2
SCHEMBL3156583 0.83 APAF1 (0.40) PTPRACYP3A4SLC7A5CPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278161-A Racemic mixtures HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
EP-0464572-A2 Aminoacid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed