SCHEMBL7433514

SCHEMBL7433514

NC(CCOc1ccncc1NC(=O)c1c[nH]c2c1C(=O)CCC2)Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 5/20 0.36
PIM3 Q86V86 3/20 0.36
PIM2 Q9P1W9 3/20 0.36
BUB1 O43683 2/20 0.34
GSK3B P49841 8/20 0.34
GSK3A P49840 2/20 0.34
ATR Q13535 4/20 0.33
MAPT P10636 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435249 0.87 BUB1 (0.35) PIM1PIM3PIM2BUB1GSK3B
SCHEMBL6093719 0.85 SGMS2 (0.37) BUB1GSK3BGSK3AMAPT
Hydrochloric Acid SCHEMBL6094797 0.85 SGMS2 (0.36) PIM1PIM3PIM2BUB1GSK3B
SCHEMBL6092102 0.84 SGMS2 (0.37) GSK3BGSK3AMAPT
SCHEMBL6094182 0.84 BUB1 (0.35) PIM1PIM3PIM2BUB1GSK3B
Hydrochloric Acid SCHEMBL6093849 0.83 SGMS2 (0.36) PIM1PIM3PIM2GSK3BGSK3A
SCHEMBL6093372 0.83 ATR (0.37) PIM1PIM3PIM2BUB1GSK3B
SCHEMBL6094276 0.82 GSK3B (0.38) PIM1PIM3PIM2BUB1GSK3B
SCHEMBL7433522 0.82 GSK3A (0.34) BUB1GSK3BGSK3AATRMAPT
SCHEMBL6094509 0.82 BUB1 (0.39) PIM1PIM3PIM2BUB1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210328-A1 FUSED PYRROLECARBOXAMIDES: A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-06-05 EP disclosed
WO-2001016103-A1 FUSED PYRROLECARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2001-03-08 WO disclosed