SCHEMBL7435249

SCHEMBL7435249

CCC(CC)CC(N)CCOc1ccncc1NC(=O)c1c[nH]c2c1C(=O)CCC2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BUB1 O43683 3/20 0.35
GSK3B P49841 9/20 0.34
ATR Q13535 6/20 0.34
MAPT P10636 4/20 0.34
PIM1 P11309 2/20 0.33
PIM3 Q86V86 2/20 0.33
PIM2 Q9P1W9 2/20 0.33
GSK3A P49840 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433514 0.87 PIM1 (0.36) BUB1GSK3BATRMAPTPIM1
SCHEMBL6093224 0.86 ATR (0.37) BUB1GSK3BATRMAPTPIM1
SCHEMBL6095690 0.85 BUB1 (0.36) BUB1GSK3BATRMAPTPIM1
SCHEMBL7392263 0.84 GSK3B (0.46) BUB1GSK3BATRMAPTGSK3A
SCHEMBL7435254 0.83 GSK3A (0.33) BUB1GSK3BATRMAPTGSK3A
SCHEMBL6095877 0.83 BUB1 (0.38) BUB1GSK3BATRMAPTPIM1
SCHEMBL6094276 0.83 GSK3B (0.38) BUB1GSK3BATRMAPTPIM1
SCHEMBL6094509 0.83 BUB1 (0.39) BUB1GSK3BATRMAPTPIM1
SCHEMBL6093349 0.82 BUB1 (0.40) BUB1GSK3BATRMAPTPIM1
Hydrochloric Acid SCHEMBL6093962 0.82 BUB1 (0.38) BUB1GSK3BATRMAPTPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210328-A1 FUSED PYRROLECARBOXAMIDES: A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-06-05 EP disclosed
WO-2001016103-A1 FUSED PYRROLECARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2001-03-08 WO disclosed