SCHEMBL7433742

SCHEMBL7433742

CC(Oc1c(Cl)cc(Cl)cc1Cl)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51
TDP1 Q9NUW8 1/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.42
PTGDR Q13258 1/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9501814 0.90 TSHR (0.58) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL2557590 0.85 ERN1 (0.45) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL2557044 0.82 TSHR (0.43) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL9780698 0.81 KMT2A (0.49) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL9780706 0.81 KMT2A (0.49) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL7788712 0.79 KMT2A (0.44) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL7788714 0.79 KMT2A (0.44) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL9780822 0.78 TDP1 (0.55) TSHRHTR2AHTR2CHTR2BTDP1
SCHEMBL1360515 0.78 TDP1 (0.55) TSHRHTR2AHTR2CHTR2BTDP1
(S)-Dichlorprop SCHEMBL1535831 0.77 TSHR (0.73) TSHRHTR2AHTR2CHTR2BPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1155010-A1 ACETAMIDO ACETONITRILE DERIVATIVES AS INHIBITORS OF CATHEPSIN L AND/OR CATHEPSIN S AstraZeneca AB (SE) 2001-11-21 EP disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000049007-A1 ACETAMIDO ACETONITRILE DERIVATIVES AS INHIBITORS OF CATHEPSIN L AND/OR CATHEPSIN S ASTRAZENECA AB (SE) 2000-08-24 WO disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed
US-4672065-A TOMATO LATE BLIGHT CHEVRON RESEARCH COMPANY (US) 1987-06-09 US disclosed
US-4535087-A FOR TOMATO LATE BLIGHT CHEVRON RESEARCH COMPANY (US) 1985-08-13 US disclosed