SCHEMBL7788714

SCHEMBL7788714

COc1c(Cl)cc(Cl)c(OC(C)C(=O)O)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
TSHR P16473 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
TPMT P51580 1/20 0.42
TDP1 Q9NUW8 1/20 0.40
ALDH1A1 P00352 6/20 0.40
HPGD P15428 2/20 0.40
KDM4E B2RXH2 4/20 0.39
GAA P10253 2/20 0.39
HSD17B10 Q99714 3/20 0.39
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
PKM P14618 1/20 0.37
CYP2C19 P33261 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
PTGDR Q13258 1/20 0.36
MAPK1 P28482 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7788712 1.00 KMT2A (0.44) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL7433742 0.79 TSHR (0.51) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL21614387 0.75 ALDH1A1 (0.42) KMT2ATSHRTPMTTDP1ALDH1A1
SCHEMBL7783284 0.75 KMT2A (0.57) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL7783289 0.75 KMT2A (0.57) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL7792299 0.75 KMT2A (0.57) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL7431492 0.74 TSHR (0.44) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL2557044 0.73 TSHR (0.43) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL9501814 0.73 TSHR (0.58) KMT2ATSHRHTR2AHTR2CHTR2B
SCHEMBL2555473 0.73 KMT2A (0.50) KMT2ATSHRHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850246-B1 PYRIMIDINE NUCLEOSIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2001-11-14 EP disclosed
EP-0850246-A2 PYRIMIDINE NUCLEOSIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1998-07-01 EP disclosed
US-5705492-A ESTERIFICATION OF PYRIMIDINE NUCLEOSIDE HOFFMANN-LA ROCHE INC. (US) 1998-01-06 US disclosed
WO-1997003082-A2 PYRIMIDINE NUCLEOSIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-01-30 WO disclosed