SCHEMBL7433850

SCHEMBL7433850

COc1cc(C(=O)C(=O)O)ccc1OCCCN1CCC(C(O)(c2ccccc2)c2ccc(F)cc2)CC1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.57
CYP2J2 P51589 3/20 0.54
HRH1 P35367 2/20 0.51
KCNH2 Q12809 2/20 0.50
ABCB11 O95342 1/20 0.50
CHRM2 P08172 1/20 0.50
HTR1A P08908 1/20 0.50
ADRA2A P08913 1/20 0.50
CHRM1 P11229 1/20 0.50
DRD2 P14416 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
DRD1 P21728 1/20 0.50
DRD4 P21917 1/20 0.50
ACHE P22303 1/20 0.50
SLC6A2 P23975 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
SLC6A4 P31645 1/20 0.50
CCKBR P32239 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437122 0.97 PAX8 (0.53) PAX8CYP2J2HRH1KCNH2ABCB11
SCHEMBL7331615 0.92 HRH1 (0.59) PAX8CYP2J2HRH1KCNH2ABCB11
SCHEMBL7442321 0.92 PAX8 (0.51) PAX8CYP2J2HRH1KCNH2ABCB11
SCHEMBL7428598 0.91 MEN1 (0.51) PAX8HRH1KCNH2ABCB11CHRM2
SCHEMBL10461477 0.90 PAX8 (0.54) PAX8CYP2J2HRH1KCNH2ABCB11
SCHEMBL6440267 0.89 ABCB11 (0.62) PAX8HRH1KCNH2ABCB11CHRM2
SCHEMBL30627531 0.89 ABCB11 (0.62) PAX8HRH1KCNH2ABCB11CHRM2
SCHEMBL7435992 0.88 HRH1 (0.54) PAX8CYP2J2HRH1KCNH2ABCB11
SCHEMBL7433635 0.87 ABCB11 (0.49) PAX8CYP2J2HRH1KCNH2ABCB11
SCHEMBL7446585 0.87 PAX8 (0.53) PAX8CYP2J2HRH1KCNH2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed