SCHEMBL7434682

SCHEMBL7434682

Oc1ccc(-c2nc3ncccc3[nH]2)cc1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.68
HPSE Q9Y251 2/20 0.65
PRMT5 O14744 3/20 0.62
PDE5A O76074 1/20 0.60
METAP1 P53582 2/20 0.57
METAP2 P50579 1/20 0.57
MGAM O43451 1/20 0.56
GAA P10253 1/20 0.56
SI P14410 1/20 0.56
MGAM2 Q2M2H8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1284270 0.84 AURKA (0.73) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL6265481 0.83 AURKA (0.68) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL28223244 0.83 AURKA (0.68) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL28693174 0.83 AURKA (0.68) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL11770396 0.83 AURKA (0.70) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL11155883 0.83 AURKA (0.67) AURKAHPSEPRMT5PDE5AMETAP1
Hydrochloric Acid SCHEMBL11776694 0.83 AURKA (0.71) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL7393911 0.83 AURKA (0.66) AURKAHPSEPRMT5PDE5AMETAP1
Hydrochloric Acid SCHEMBL11772488 0.82 AURKA (0.66) AURKAHPSEPRMT5PDE5AMETAP1
SCHEMBL1170747 0.82 METAP1 (0.72) AURKAHPSEPRMT5PDE5AMETAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001066526-A1 ESTER DERIVATIVES OF DIMETHYLPROPIONIC ACID AND PHARMACETUICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2001-09-13 WO disclosed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP disclosed
US-3985891-A CARDIOTONICS, ANTICOAGULANTS BOEHRINGER INGELHEIM GMBH (DT) 1976-10-12 US disclosed