SCHEMBL28693174

SCHEMBL28693174

Clc1ccc(-c2nc3ncccc3[nH]2)cc1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.68
HPSE Q9Y251 2/20 0.61
PRMT5 O14744 3/20 0.58
METAP1 P53582 2/20 0.57
METAP2 P50579 1/20 0.57
MGAM O43451 1/20 0.56
GAA P10253 1/20 0.56
SI P14410 1/20 0.56
MGAM2 Q2M2H8 1/20 0.56
TP53 P04637 1/20 0.54
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
PDE5A O76074 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11772488 0.98 AURKA (0.66) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL3925926 0.91 AURKA (0.68) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL1284270 0.84 AURKA (0.73) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL28223244 0.83 AURKA (0.68) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL6265481 0.83 AURKA (0.68) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL7434682 0.83 AURKA (0.68) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL11770396 0.83 AURKA (0.70) AURKAHPSEPRMT5METAP1METAP2
Hydrochloric Acid SCHEMBL11776694 0.83 AURKA (0.71) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL11155883 0.83 AURKA (0.67) AURKAHPSEPRMT5METAP1METAP2
SCHEMBL23870533 0.83 AURKA (0.65) AURKAHPSEPRMT5METAP1METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113956208-B Aryl heterocyclic derivative and synthesis method thereof 郑州大学 2023-08-15 CN disclosed
CN-113956208-A Aryl heterocyclic derivative and synthetic method thereof 郑州大学 2022-01-21 CN disclosed